Preface (B.E. Maryanoff, A.B. Reitz).
Novel peptide mimetic building blocks and strategies for efficient lead finding (D. Obrecht et al.).
Recent advances in the medicinal chemistry of taxoid anticancer agents (I. Ojima et al.). Synthesis and structure-activity relationships of peroxidic antimalarials based on artemisinin (M.A. Avery et al.).
Design of compound libraries for detecting and pursuing novel small molecule leads (A.M. Ferguson, R.D. Cramer).
A theoretical model of the human thrombin receptor (PAR-1), the first known protease-activated G-protein-coupled receptor (M.P. Beavers et al.).
Farnesyl transferase inhibitors: design of a new class of cancer chemotherapeutic agents (T.M. Williams, C.J. Dinsmore).